Selective Alkylation of Ambient 5-Halopyrimidin-2-one Anion.
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چکیده
منابع مشابه
Studies on the Alkylation of Quinolin-2(1h)-one Derivatives
Alkylation of quinolin-2(1H)-one (1) and its C(6) and C(7) substituted dervatives (OMe, OBn, and Cl) with 2-bromoacetophenone or chloroacetone under basic condition (K2CO3 in DMF) gave a mixture of N1and O2alkylated products with the former one as a major product. However, alkylation of 8-methoxy-, 8-benzyloxy-, and 8-chloroquinolin-2(1H)-ones under the same reaction conditions gave exclusively...
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ژورنال
عنوان ژورنال: Acta Chemica Scandinavica
سال: 1981
ISSN: 0904-213X
DOI: 10.3891/acta.chem.scand.35b-0069